Varenicline-15N,13C, d2
Varenicline-15N,13C, d2
SKU:QM-0079142
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Product Details
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Description
Varenicline-15N,13C, d2 is 15N and deuterated labeled Varenicline. Varenicline (CP 526555) is an orally active partial agonist of α4β2 nicotinic acetylcholine receptor (α4β2 nAChR, IC50=250 nM), which is the principal mediator of nicotine dependence. Varenicline is also a partial agonist of α6β2 nAChR and a full agonist of α7β2 nAChR. Varenicline blocks the direct agonist effects of nicotine on nAChR while stimulates nAChR in a more moderate way, being widely used as an aid of smoking cessation[1][2][3][4][5].
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Molecular Formula
C12 13CH11D2N2 15N
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Molecular Weight
215.26
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Smiles
[2H]C1([2H])[15NH][13CH2]C2CC1C3=C2C=C4N=CC=NC4=C3
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Target
Isotope-Labeled Compounds; nAChR
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Solubility
10 mM in DMSO
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Shipping Conditions
Room temperature
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Varenicline-15N,13C, d2
Varenicline-15N,13C, d2 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.