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Varenicline-15N3 (hydrochloride) [CAS 1244134-80-2]

Varenicline-15N3 (hydrochloride) [CAS 1244134-80-2]

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SKU:QM-0079151

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  • Description

    Varenicline-15N3 Hydrochloride (CP 526555-15N3 Hydrochloride) is the 15N labeled isotope of Varenicline hydrochloride. Varenicline (CP 526555) is an orally active partial agonist of α4β2 nicotinic acetylcholine receptor (α4β2 nAChR, IC50 = 250 nM), which is the principal mediator of nicotine dependence. Varenicline is also a partial agonist of α6β2 nAChR and a full agonist of α6β2 nAChR. Varenicline blocks the direct agonist effects of nicotine on nAChR while stimulates nAChR in a more moderate way, being widely used as an aid of smoking cessation[1][2][3][4][5].

  • CAS Number

    [1244134-80-2]

  • Molecular Formula

    C13H14Cl 15N3

  • Molecular Weight

    250.7

  • Smiles

    C1(C2CC3C[15NH]C2)=C3C=C([15N]=CC=[15N]4)C4=C1.Cl

  • Target

    Isotope-Labeled Compounds; nAChR

  • Shipping Conditions

    Room temperature

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Varenicline-15N3 (hydrochloride) [CAS 1244134-80-2]

Varenicline-15N3 (hydrochloride) is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.