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VP3.15 (dihydrobromide) [CAS 1281681-33-1]

VP3.15 (dihydrobromide) [CAS 1281681-33-1]

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SKU:QM-0142682-01

£118.38 GBP
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  • Description

    VP3.15 dihydrobromide is a potent, orally bioavailable and CNS-penetrant dual phosphodiesterase (PDE) 7- glycogen synthase kinase (GSK) 3 inhibitor, with IC50s of 1.59 μM and 0.88 μM for PDE7 and GSK-3, respectively. VP3.15 dihydrobromide has neuroprotective and neuroreparative activities, thus as potential combined anti-inflammatory and pro-remyelinating therapies for multiple sclerosis (MS) [1].

  • CAS Number

    [1281681-33-1]

  • Molecular Formula

    C20H24Br2N4OS

  • Molecular Weight

    528.3

  • Smiles

    [H]Br.[H]Br.N1(CC/N=C2N=C(C3=CC=CC=C3)N(C4=CC=CC=C4)S/2)CCOCC1

  • Target

    GSK-3; Phosphodiesterase (PDE)

  • Isoform

    PDE7

  • Purity

    98.01

  • Solubility

    DMSO : 62.5 mg/mL (ultrasonic)

  • Storage Conditions

    4°C (Powder, sealed storage, away from moisture)

  • Shipping Conditions

    Room Temperature

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Variant Variant total Quantity Price Variant total
5 mgQM-0142682-01
5 mgQM-0142682-01
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10 mM - 1 mLQM-0142682-02
10 mM - 1 mLQM-0142682-02
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10 mgQM-0142682-03
10 mgQM-0142682-03
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25 mgQM-0142682-04
25 mgQM-0142682-04
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50 mgQM-0142682-05
50 mgQM-0142682-05
£664.79/ea
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100 mgQM-0142682-06
100 mgQM-0142682-06
£1,116.77/ea
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VP3.15 (dihydrobromide) [CAS 1281681-33-1]

VP3.15 (dihydrobromide) is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.