Y-29794 (tosylate) [CAS 143984-17-2]
Y-29794 (tosylate) [CAS 143984-17-2]
SKU:QM-0132112-01
Couldn't load pickup availability
Request quote or documents
![Y-29794 (tosylate) [CAS 143984-17-2]](http://quantimol.com/cdn/shop/files/quantimol-021.png?v=1773515276&width=1445)
Product Details
-
Description
Y-29794 tosylate is a selective, orally active inhibitor for non-peptide prolyl endopeptidase (PREP), with an IC50 of 3 nM and a Ki of 0.95 nM. Y-29794 tosylate enhances the effect of thyrotropin-releasing hormone (TRH) on the release of ACh in the rat hippocampus, exhibits potential neuroprotective efficacy. Y-29794 tosylate exhibits anticancer activity through inhibition of the IRS1-AKT-mTORC1 pathway. Y-29794 tosylate penetrates the brain-blood barrier (BBB) [1][2].
-
CAS Number
[143984-17-2]
-
Molecular Formula
C30H42N2O4S3
-
Molecular Weight
590.86
-
Smiles
O=C(C1=CC=C(C(C)C)N=C1SCCCCCCCCN(C)C)C2=CC=CS2.O=S(C3=CC=C(C)C=C3)(O)=O
-
Target
Prolyl Endopeptidase (PREP)
-
Isoform
PREP
-
Solubility
10 mM in DMSO
-
Shipping Conditions
Room temperature
Related Products
- QM-0053803 γ-Linolenic acid ethyl ester-d5
- QM-0052686-01 β-Phenyl GHB (sodium) [CAS 40951-19-7]
- QM-0052524 β-Nicotinamide mononucleotide, reduced form (disodium) (Standard) [CAS 108347-85-9]
- QM-0052354-01 ω-azido-C6 Ceramide [CAS 2108102-18-5]
- QM-0051720-01 β-Phenylethyl β-D-glucoside [CAS 18997-54-1]
- QM-0048489-01 β-N-methylamino-L-alanine (hydrochloride) (Standard) [CAS 16012-55-8]
- QM-0022874 β-Prumycin hydrochloride [CAS 54612-74-7]
- QM-0206006 β-Nicotinamide adenine dinucleotide reduced (dipotassium) [CAS 104809-32-7]
- QM-0204726-01 β-Nicotinamide mononucleotide, reduced form (disodium) [CAS 108347-85-9]
- QM-0204366-01 β-N-methylamino-L-alanine (hydrochloride) [CAS 16012-55-8]
Other industry favorites
- QM-0053803 γ-Linolenic acid ethyl ester-d5
- QM-0052686-01 β-Phenyl GHB (sodium) [CAS 40951-19-7]
- QM-0054913 β-D-Galactopyranose,2,3,4,6-tetrakis-O- (phenylmethyl),1-acetate [CAS 3866-62-4]
- QM-0054858-01 α-D-Mannopyranosyl chloride, 2,3,4,6-tetraacetate [CAS 14257-40-0]
- QM-0016946-01 β-Carboline-1-carboxylic acid [CAS 26052-96-0]
- QM-0016203 β-D-Glu-benzylalcohol-di (amide-C2) -mal
- QM-0178574-01 β-Sitosterol acetate, 40% (contains Campesterol acetate) [CAS 915-05-9]
- QM-0168310-01 γ-Linolenyl alcohol [CAS 24149-05-1]
- QM-0050582 β-D-Galaltosamine (hydrochloride) [CAS 14257-79-5]
- QM-0049152-01 β-keto Phentermine (hydrochloride) [CAS 6946-08-3]
Y-29794 (tosylate) [CAS 143984-17-2]
Y-29794 (tosylate) is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.