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σ1 Receptor/μ Opioid receptor modulator 2 [CAS 3009018-61-2]
σ1 Receptor/μ Opioid receptor modulator 2 [CAS 3009018-61-2]
SKU:QM-0073595
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Product Details
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Description
σ1 Receptor/μ Opioid receptor modulator 2 (compound 4x) is a dual μOR agonist/σ1R antagonist, and displays picomolar μOR agonism activity (EC50: 0.6 ± 0.2 nM) and good σ1R inhibitory activity (Ki: 363.7 ± 5.6 nM) . σ1 Receptor/μ Opioid receptor modulator 2 exhibits robust analgesic effects in various pain models[1].
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CAS Number
[3009018-61-2]
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Molecular Formula
C23H31N3O
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Molecular Weight
365.51
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Smiles
O=C(N(C1=CC=CC=N1)CC(N2CCC(CC2)C3=CC=CC=C3)CC)CC
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Target
Opioid Receptor; Sigma Receptor
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Solubility
10 mM in DMSO
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Shipping Conditions
Room temperature
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σ1 Receptor/μ Opioid receptor modulator 2 [CAS 3009018-61-2]
σ1 Receptor/μ Opioid receptor modulator 2 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.