Navafenterol (saccharinate) [CAS 1648550-37-1]
Navafenterol (saccharinate) [CAS 1648550-37-1]
SKU:QM-0059902
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Product Details
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Description
Navafenterol (AZD-8871) saccharinate is an inhaled dual-acting, potent, selective, and long-lasting M3-antagonist/β2-agonist (MABA) with long-lasting effects and favorable safety profile. The pIC50 is 9.5 for human M3 receptor, and the pEC50 is 9.5 for β2-adrenoceptor. Navafenterol saccharinate can be used for the research of chronic obstructive pulmonary disease (COPD) . Bronchoprotective and antisialagogue effects. Favorable cardiovascular profile[1].
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CAS Number
[1648550-37-1]
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Molecular Formula
C45H47N7O9S3
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Molecular Weight
926.09
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Smiles
O=C(C(O)(C1=CC=CS1)C2=CC=CS2)O[C@H]3CC[C@@H](CC3)N(C)CCCN4N=NC5=CC(CNC[C@H](O)C6=CC=C(C7=C6C=CC(N7)=O)O)=CC=C54.O=S8(C9=CC=CC=C9C(N8)=O)=O
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Target
Adrenergic Receptor; mAChR
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Isoform
MAChR3
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Solubility
10 mM in DMSO
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Shipping Conditions
Room temperature
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Navafenterol (saccharinate) [CAS 1648550-37-1]
Navafenterol (saccharinate) is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.