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5-HT2CR agonist 1 [CAS 1216074-15-5]
5-HT2CR agonist 1 [CAS 1216074-15-5]
SKU:QM-0072932
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Product Details
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Description
5-HT2CR agonist 1 (compound 8), a 7-chloro analogue, is a selective 5-HT2CR partial agonist (Emax=71.09%) with an EC50 value of 121.5 nM and no observed activity toward 5-HT2AR or 5-HT2BR. 5-HT2CR agonist 1 exhibits no recruitment activity for β-arrestin and shows low inhibition of hERG at 10 μM[1].
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CAS Number
[1216074-15-5]
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Molecular Formula
C13H14ClNO
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Molecular Weight
235.71
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Smiles
ClC1=CC=C2C=CC3(OC2=C1)CCNCC3
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Target
5-HT Receptor
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Isoform
α-1 microglobulin
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Solubility
10 mM in DMSO
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Shipping Conditions
Room temperature
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5-HT2CR agonist 1 [CAS 1216074-15-5]
5-HT2CR agonist 1 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.