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5-HT6R antagonist 3
5-HT6R antagonist 3
SKU:QM-0073657
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Product Details
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Description
5-HT6R antagonist 3 (compound 15) is a potent, selective and brain-penetrant 5-HT6R antagonist with Ki values of 14 nM, 3533 nM, 35 nM, 1449 nM for 5-HT6, 5-HT1A, 5-HT2A, 5-HT7, respectively. 5-HT6R antagonist 3 shows anxiolytic-like and properties neuroprotective and procognitive-like effects. 5-HT6R antagonist 3 has the potential for the research of Alzheimer’s Disease[1].
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Molecular Formula
C21H26N6Se
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Molecular Weight
441.43
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Smiles
CC(C)([Se]C1=CC2=C(C=C1)C=CC=C2)C3=NC(N4CCN(CC4)C)=NC(N)=N3
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Target
5-HT Receptor
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Isoform
5-HT1 Receptor;5-HT2 Receptor;5-HT7 Receptor; mLAG-3; MUC2; MUC3; α-1 microglobulin
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Solubility
10 mM in DMSO
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Shipping Conditions
Room temperature
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5-HT6R antagonist 3
5-HT6R antagonist 3 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.