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A2AR/A2BR antagonist 1
A2AR/A2BR antagonist 1
SKU:QM-0086676
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Product Details
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Description
A2AR/A2BR antagonist 1 (compound 7ai) has a dual antagonistic effect on A2AR/A2BR, with the IC50 values of 11.2 nM and 6.4 nM for A2AR and A2BR, respectively. A2AR/A2BR antagonist 1 promotes T cell-mediated cancer cell death[1].
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Molecular Formula
C24H17N9
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Molecular Weight
431.45
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Smiles
NC1=NC(C2=CN(N=N2)CC3=CNC4=C3C=C(C=C4)C#N)=CC(C5=CC=CC(C#N)=C5C)=N1
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Target
Adenosine Receptor
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Isoform
Adenosine A2A receptor (A2AR) ; Adenosine A2B receptor (A2BR)
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Solubility
10 mM in DMSO
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Shipping Conditions
Room temperature
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A2AR/A2BR antagonist 1
A2AR/A2BR antagonist 1 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.