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Adenosine receptor antagonist 5
Adenosine receptor antagonist 5
SKU:QM-0126299
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Product Details
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Description
Adenosine receptor antagonist 5 (Compound 39) is a selective antagonist for human adenosine A3 receptor (hA3R) with Ki of 12 nM. Adenosine receptor antagonist 5 inhibits IB-MECA -induced cAMP accumulation in NCI-H1792 cell, inhibits the proliferation of cancer cell LK-2 and NCI-H1792. Adenosine receptor antagonist 5 exhibits a fast metabolic rate in human liver microsomes[1].
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Molecular Formula
C17H11BrCl2N4O3
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Molecular Weight
470.1
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Smiles
CC1=C(C(C2=C(C=CC=C2Cl)Cl)=NO1)C(O/N=C(C3=CC=C(C=N3)Br)\N)=O
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Target
Adenosine Receptor
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Isoform
Adenosine A3 receptor (A3R)
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Shipping Conditions
Room temperature
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Adenosine receptor antagonist 5
Adenosine receptor antagonist 5 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.