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APJ antagonist-1
APJ antagonist-1
SKU:QM-0013439
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Product Details
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Description
APJ antagonist-1 is an apelin receptor (APJ) antagonist. APJ antagonist-1 shows strong β-arrestin inhibition with an IC50 of 3.1 μM. APJ antagonist-1 selectively inhibits APJ-overexpressing cancer cells and suppresses apelin-induced endothelial cell migration. APJ antagonist-1exhibits high metabolic stability. APJ antagonist-1 can used for the studies of ovarian cancer and tumor angiogenesis[1].
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Molecular Formula
C18H15N3O6S2
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Molecular Weight
433.46
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Smiles
O=S(C1=CC=C([N+]([O-])=O)C=C1)(OC2=CC(CSC3=NC=CC=N3)=CC=C2OC)=O
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Target
Apelin Receptor (APJ)
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Shipping Conditions
Room temperature
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APJ antagonist-1
APJ antagonist-1 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.