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APJ receptor agonist 1 [CAS 2287153-38-0]
APJ receptor agonist 1 [CAS 2287153-38-0]
SKU:QM-0062086
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Product Details
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Description
APJ receptor agonist 1, a biphenyl acid derivative, is a potent APJ receptor (APJ-R) agonist (EC50s 0.093 and 0.12 nM for human and rat APJ-R, respectively) . APJ receptor agonist 1 displays in vitro potency to apelin-13, the endogenous peptidic ligand for the APJ receptor. APJ receptor agonist 1 has the potential for the research of heart failure[1].
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CAS Number
[2287153-38-0]
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Molecular Formula
C31H26ClN3O3
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Molecular Weight
524.01
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Smiles
O=C(C1=CC(C(N[C@@H](C2=CC=CC=C2)CCC)=O)=CC=[C@]1[C@]3=C(Cl)C=CC=C3C4=NC5=CC=CC=C5N4)O
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Target
Apelin Receptor (APJ)
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Solubility
10 mM in DMSO
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Shipping Conditions
Room temperature
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APJ receptor agonist 1 [CAS 2287153-38-0]
APJ receptor agonist 1 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.