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APJ receptor agonist 5 [CAS 2135514-20-2]

APJ receptor agonist 5 [CAS 2135514-20-2]

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QM-0066163-01

£464.31 GBP
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Product Details

  • Description

    APJ receptor agonist 5 (compound 3) is a potent and orally active agonist of apelin receptor (APJ) with an EC50 of 0.4 nM. APJ receptor agonist 5 displays excellent pharmacokinetic profiles in the rodent heart failure (HF) model. APJ receptor agonist 5 also shows an acceptable safety profile in preclinical toxicology studies. APJ receptor agonist 5 leads to improved cardiac function and can be used for researching the HF disease[1].

  • CAS Number

    [2135514-20-2]

  • Molecular Formula

    C26H29N3O6

  • Molecular Weight

    479.52

  • Smiles

    CCOCC(N(C1=C(C=CC=C1OC)OC)C(O)=C2C(N3C[C@](C4=CC=CC=C4)([H])CC3)=O)=NC2=O

  • Target

    Apelin Receptor (APJ)

  • Solubility

    10 mM in DMSO

  • Shipping Conditions

    Room temperature
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Variant Variant total Quantity Price Variant total
5 mgQM-0066163-01
5 mgQM-0066163-01
£464.31/ea		 £0.00
£464.31/ea £0.00
10 mgQM-0066163-02
10 mgQM-0066163-02
£727.97/ea		 £0.00
£727.97/ea £0.00
25 mgQM-0066163-03
25 mgQM-0066163-03
£1,305.10/ea		 £0.00
£1,305.10/ea £0.00
50 mgQM-0066163-04
50 mgQM-0066163-04
£2,058.39/ea		 £0.00
£2,058.39/ea £0.00
100 mgQM-0066163-05
100 mgQM-0066163-05
£3,313.49/ea		 £0.00
£3,313.49/ea £0.00
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APJ receptor agonist 5 [CAS 2135514-20-2]

APJ receptor agonist 5 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.