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AT1R antagonist 3 [CAS 3053482-15-5]
AT1R antagonist 3 [CAS 3053482-15-5]
SKU:QM-0098654
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Product Details
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Description
AT1R antagonist 3 (Compound 1) is an antagonist for angiotensin II type 1 receptor (AT1R) and an inhibitor for calcium channel type-L CaV1.2 (IC50=0.57 μM) . AT1R antagonist 3 exhibits vasodilation efficacy in solated rat aorta (10 μM, 88.7%) and antihypertensive efficacy in rat models[1].
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CAS Number
[3053482-15-5]
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Molecular Formula
C22H16N6O2S
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Molecular Weight
428.47
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Smiles
O=C(C1=CC2=C(NC(SCC3=CC=C(C=C3)C4=C(C=CC=C4)C5=NN=NN5)=N2)C=C1)O
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Target
Angiotensin Receptor; Calcium Channel
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Isoform
L-type calcium channel
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Shipping Conditions
Room temperature
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AT1R antagonist 3 [CAS 3053482-15-5]
AT1R antagonist 3 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.