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AT2R antagonist 1 [CAS 2709031-17-2]
AT2R antagonist 1 [CAS 2709031-17-2]
SKU:QM-0066848
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Product Details
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Description
AT2R antagonist 1 (compound 21) is a potent and high selective AT2R (angiotensin II AT2 receptor) ligand. AT2R antagonist 1 exhibits a fair AT2R affinity, with a Ki of 29 nM. AT2R antagonist 1 also inhibits common agent-metabolizing CYP enzymes. AT2R antagonist 1 shows high stability in human, rat and mouse liver microsomes[1].
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CAS Number
[2709031-17-2]
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Molecular Formula
C23H30N4O4S2
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Molecular Weight
490.64
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Smiles
COC(NS(=O)(C1=C(N=C(S1)CC(C)C)C2=CC=C(C=C2)CN3C=CN=C3C(C)(C)C)=O)=O
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Target
Angiotensin Receptor
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Isoform
AT2 Receptor
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Solubility
10 mM in DMSO
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Shipping Conditions
Room temperature
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AT2R antagonist 1 [CAS 2709031-17-2]
AT2R antagonist 1 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.