1 1

Aurora-A ligand 1 [CAS 2541626-73-5]

Aurora-A ligand 1 [CAS 2541626-73-5]

Size

QM-0008496-01

£282.06 GBP
Sale Sold out

Request quote or documents

View full details

Product Details

  • Description

    Aurora-A ligand 1 is a high-affinity and specific Aurora-A inhibitor with a dissociation constant (Kd) value of 0.85 nM. Aurora-A ligand 1 can serve as a ligand for target protein (Ligands for Target Protein for PROTAC) for the development of PROTAC Aurora-A degraders with antitumor activity. Aurora-A ligand 1 can be used for the synthesis of HLB-0532259. HLB-0532259 shows anti-tumor activity against neuroblastoma[1].

  • CAS Number

    [2541626-73-5]

  • Molecular Formula

    C21H23N5O3

  • Molecular Weight

    393.44

  • Smiles

    O=C(N(C)C)C(N1C2CCCC2)=CC3=C1N=C(NC4=CC=C(C(O)=O)C=C4)N=C3

  • Target

    Aurora Kinase; Ligands for Target Protein for PROTAC

  • Concentration

    10mM

  • Purity

    98.75

  • Solubility

    DMSO : 100 mg/mL (ultrasonic)

  • Storage Conditions

    -20°C, 3 years; 4°C, 2 years (Powder)

  • Shipping Conditions

    Room Temperature
Learn more
Variant Variant total Quantity Price Variant total
5 mgQM-0008496-01
5 mgQM-0008496-01
£171.90
£282.06/ea
 £0.00
£171.90
£282.06/ea
 £0.00
10 mM - 1 mLQM-0008496-02
10 mM - 1 mLQM-0008496-02
£189.00
£305.15/ea
 £0.00
£189.00
£305.15/ea
 £0.00
10 mgQM-0008496-03
10 mgQM-0008496-03
£274.50
£420.57/ea
 £0.00
£274.50
£420.57/ea
 £0.00
25 mgQM-0008496-04
25 mgQM-0008496-04
£549.00
£791.15/ea
 £0.00
£549.00
£791.15/ea
 £0.00
50 mgQM-0008496-05
50 mgQM-0008496-05
£882.90
£1,241.91/ea
 £0.00
£882.90
£1,241.91/ea
 £0.00
View cart
0

Total items

£0.00

Product subtotal

Taxes, discounts and shipping calculated at checkout.
View cart

Related Products

Other industry favorites

Aurora-A ligand 1 [CAS 2541626-73-5]

Aurora-A ligand 1 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.