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BET bromodomain inhibitor 1 [CAS 2411226-02-1]

BET bromodomain inhibitor 1 [CAS 2411226-02-1]

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QM-0077811-01

£265.06 GBP
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Product Details

  • Description

    BET bromodomain inhibitor 1 is an orally active, selective bromodomain and extra-terminal (BET) bromodomain inhibitor with an IC50 of 2.6 nM for BRD4. BET bromodomain inhibitor 1 binds to BRD2 (2), BRD3 (2), BRD4 (1), BRD4 (2), and BRDT (2) with high affinities (Kd values of 1.3 nM, 1.0 nM, 3.0 nM, 1.6 nM, 2.1 nM, respectively) . bromodomain inhibitor 1 has anti-cancer activity[1].

  • CAS Number

    [2411226-02-1]

  • Molecular Formula

    C22H19F2N3O4S

  • Molecular Weight

    459.47

  • Smiles

    O=C1C2=C(C)C=C(C3=CC(CS(=O)(CC)=O)=CN=C3OC4=CC=C(F)C=C4F)N2C=CN1

  • Target

    Epigenetic Reader Domain

  • Isoform

    BRD2; BRD3; BRD4; BRDT

  • Purity

    99.91

  • Solubility

    DMSO : 100 mg/mL (ultrasonic; warming; heat to 60°C)

  • Storage Conditions

    -20°C, 3 years; 4°C, 2 years (Powder)

  • Shipping Conditions

    Room Temperature
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Variant Variant total Quantity Price Variant total
5 mgQM-0077811-01
5 mgQM-0077811-01
£265.06/ea		 £0.00
£265.06/ea £0.00
10 mM - 1 mLQM-0077811-02
10 mM - 1 mLQM-0077811-02
£267.49/ea		 £0.00
£267.49/ea £0.00
10 mgQM-0077811-03
10 mgQM-0077811-03
£395.06/ea		 £0.00
£395.06/ea £0.00
25 mgQM-0077811-04
25 mgQM-0077811-04
£740.12/ea		 £0.00
£740.12/ea £0.00
50 mgQM-0077811-05
50 mgQM-0077811-05
£1,120.41/ea		 £0.00
£1,120.41/ea £0.00
100 mgQM-0077811-06
100 mgQM-0077811-06
£1,658.66/ea		 £0.00
£1,658.66/ea £0.00
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BET bromodomain inhibitor 1 [CAS 2411226-02-1]

BET bromodomain inhibitor 1 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.