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BRD4 Inhibitor-28 [CAS 2468960-80-5]
BRD4 Inhibitor-28 [CAS 2468960-80-5]
SKU:QM-0068424
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Product Details
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Description
BRD4 Inhibitor-28 (Compound 18) is an orally active BRD4 Inhibitor. BRD4 Inhibitor-28 inhibits BRD40-BD1, BRD40-BD2 with IC50s of 15, 55 nM. BRD4 Inhibitor-28 also inhibits BRD2-BD1, BRD3-BD1, BRDT-BD1 with IC50s of 19, 25, 68 nM. BRD4 Inhibitor-28 has anti-melanoma activity[1].
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CAS Number
[2468960-80-5]
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Molecular Formula
C23H21N3O3
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Molecular Weight
387.43
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Smiles
O=C1N2CCOC3=C2C(N1CC4=CC=CC=C4)=CC(C5=CN(C(C(C)=C5)=O)C)=C3
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Target
Epigenetic Reader Domain
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Solubility
10 mM in DMSO
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Shipping Conditions
Room temperature
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BRD4 Inhibitor-28 [CAS 2468960-80-5]
BRD4 Inhibitor-28 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.