BRM/BRG1 ATP Inhibitor-1 [CAS 2270879-17-7]
BRM/BRG1 ATP Inhibitor-1 [CAS 2270879-17-7]
SKU:QM-0139596-01
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Product Details
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Description
BRM/BRG1 ATP Inhibitor-1 (compound 14) is an orally active allosteric dual brahma homolog (BRM) /SWI/SNF related matrix associated actin dependent regulator of chromatin subfamily A member 2 (SMARCA2) and brahma related gene 1 (BRG1) /SMARCA4 ATPase activity inhibitor, both IC50s are below 0.005 µM. BRM/BRG1 ATP Inhibitor-1 has anticancer activity[1].
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CAS Number
[2270879-17-7]
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Molecular Formula
C11H9F3N4O2S
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Molecular Weight
318.27
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Smiles
FC1=CC(NC(NC2=CC(C(F)F)=NS2)=O)=C(CO)C=N1
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Target
Epigenetic Reader Domain
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Purity
99.72
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Solubility
DMSO : 200 mg/mL (ultrasonic; warming; heat to 60°C)
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Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
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Shipping Conditions
Room Temperature
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BRM/BRG1 ATP Inhibitor-1 [CAS 2270879-17-7]
BRM/BRG1 ATP Inhibitor-1 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.