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CB1/2 agonist 4 [CAS 2772949-38-7]
CB1/2 agonist 4 [CAS 2772949-38-7]
SKU:QM-0068768
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Product Details
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Description
CB1/2 agonist 4 is a full CB1 agonist and CB2 partial agonist with EC50 values of 15.09 nM and 1.16 nM, respectively. CB1/2 agonist 4 also has hCB1 and hCB2 receptor affinities with Ki values of 1.1 nM and 4.2 nM, respectively. CB1/2 agonist 4 has a significant antinociceptive activity, and also can activate cannabinoid and TRPV1 receptor with values of IC50 and EC50 is 0.8 μM and 0.12 μM, respectively[1].
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CAS Number
[2772949-38-7]
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Molecular Formula
C27H45NO3
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Molecular Weight
431.65
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Smiles
O=C(NC1CC1)CCCCCCCOC2=CC(C(CCCCCC)(C)C)=CC(OC)=C2
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Target
Cannabinoid Receptor
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Solubility
10 mM in DMSO
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Shipping Conditions
Room temperature
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CB1/2 agonist 4 [CAS 2772949-38-7]
CB1/2 agonist 4 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.