CB2R antagonist 3
CB2R antagonist 3
SKU:QM-0150852-01
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Product Details
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Description
CB2R antagonist 3 is a selective antagonist of cannabinoid type 2 receptor (CB2R). CB2R antagonist 3 has high affinity for human CB2R and specific selectivity for CB1R. CB2R antagonist 3 can be combined with CB65 , the activator of CB2R. CB2R antagonist 3 effectively up-regulates the expression of anti-inflammatory cytokines and down-regulates the expression of pro-inflammatory cytokines[1].
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Molecular Formula
C27H42N2O
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Molecular Weight
410.64
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Smiles
CCCCCNC1=C(C=C(C=C1)CCCCC)C(NC23CC4CC(C3)CC(C2)C4)=O
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Target
Cannabinoid Receptor
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Isoform
CB2
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Purity
98.08
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Solubility
DMSO : 100 mg/mL (ultrasonic; warming; heat to 60°C)
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Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
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Shipping Conditions
Room Temperature
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CB2R antagonist 3
CB2R antagonist 3 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.