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ERα antagonist 2
ERα antagonist 2
SKU:QM-0015884
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Product Details
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Description
ERα antagonist 2 (Compound 5b) is an ER-α antagonist with an IC50 value of 1729 nM. ERα antagonist 2 exhibits significant inhibitory activity against breast cancer cell lines, and is still effective against ER-negative cells (MDA-MB-231), suggesting the existence of ER-independent pathways. ERα antagonist 2 can be used for the study of breast cancer[1].
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Molecular Formula
C46H38N6O4S2
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Molecular Weight
802.96
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Smiles
CC(C=C1)=CC=C1S(N(C(C2=CN(CC3=CC=CC=C3)C4=C2C=CC=C4)=NN5S(C6=CC=C(C)C=C6)(=O)=O)N=C5C7=CN(C8=C7C=CC=C8)CC9=CC=CC=C9)(=O)=O
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Target
Estrogen Receptor/ERR
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Isoform
ERα
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Shipping Conditions
Room temperature
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ERα antagonist 2
ERα antagonist 2 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.