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ERK1/2 inhibitor 1 [CAS 2095719-90-5]
ERK1/2 inhibitor 1 [CAS 2095719-90-5]
SKU:QM-0137439-01
£376.83 GBP
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Product Details
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Description
ERK1/2 inhibitor 1 is a potent, orally bioavailable ERK1/2 inhibitor, showing 60% inhibition at 1 nM and an IC50 of 3.0 nM against ERK1 and ERK2, respectively[1].
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CAS Number
[2095719-90-5]
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Molecular Formula
C29H32ClN5O4
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Molecular Weight
550.05
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Smiles
ClC1=CN=C(NC2CCOCC2)N=C1C3=CC=C(CN([C@H](C)C(N[C@H](CO)C4=CC=CC(C)=C4)=O)C5=O)C5=C3
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Target
ERK
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Isoform
ERK1; ERK2
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Concentration
10mM
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Purity
99.58
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Solubility
DMSO : 250 mg/mL (ultrasonic)
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Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
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Shipping Conditions
Room Temperature
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ERK1/2 inhibitor 1 [CAS 2095719-90-5]
ERK1/2 inhibitor 1 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.