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Estrogen receptor modulator 8 [CAS 2170766-56-8]
Estrogen receptor modulator 8 [CAS 2170766-56-8]
SKU:QM-0070737
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Product Details
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Description
Estrogen receptor modulator 8 (Compound 4) down-regulates estrogen receptor with an IC50 of 0.1 nM-10 nM. Estrogen receptor modulator 8 degrades ERα (IC50: 25.7 nM in vitro, 0.136 nM in MCF-7 cell) . Estrogen receptor modulator 8 also inhibits MCF-7 cell growth (IC50: 0.1 nM), and MCF-7 tumor growth[1].
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CAS Number
[2170766-56-8]
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Molecular Formula
C25H24F4N2O2
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Molecular Weight
460.46
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Smiles
CC(C)(F)CN1[C@H](C2=C(C=C(C=C2F)/C=C/C(O)=O)F)C3=C(C[C@H]1C)C4=C(F)C=CC=C4N3
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Target
Estrogen Receptor/ERR
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Solubility
10 mM in DMSO
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Shipping Conditions
Room temperature
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Estrogen receptor modulator 8 [CAS 2170766-56-8]
Estrogen receptor modulator 8 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.