G-Protein antagonist peptide (TFA)
G-Protein antagonist peptide (TFA)
SKU:QM-0172964-01
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Product Details
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Description
G-Protein antagonist peptide TFA is a truncated substance P-related peptide, competes with receptor for G protein binding. G-Protein antagonist peptide TFA inhibits the activation of Gi or Go by M2 muscarinic cholinergic receptor (M2 mAChR) or of Gs by beta-adrenergic receptor in the reconstituted phospholipid vesicles, assayed by receptor-promoted GTP hydrolysis[1].
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Molecular Formula
C59H65F3N12O11S
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Molecular Weight
1207.28
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Smiles
CSCC[C@@H](C(N)=O)NC([C@@H](CC1=CNC2=C1C=CC=C2)NC([C@@H](CC3=CNC4=C3C=CC=C4)NC([C@H](CC5=CC=CC=C5)NC([C@@H](CC6=CNC7=C6C=CC=C7)NC([C@H](CCC(N)=O)NC([C@H](CC8)NC8=O)=O)=O)=O)=O)=O)=O.O=C(O)C(F)(F)F
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Target
Adrenergic Receptor; mAChR
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Isoform
MAChR2
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Purity
97.07
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Solubility
DMSO : 100 mg/mL (ultrasonic)
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Storage Conditions
-80°C, 2 years; -20°C, 1 year (Powder, stored under nitrogen, away from moisture)
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Shipping Conditions
Blue Ice
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G-Protein antagonist peptide (TFA)
G-Protein antagonist peptide (TFA) is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.