GABAA receptor modulator-10
GABAA receptor modulator-10
SKU:QM-0013337
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Product Details
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Description
GABAA receptor modulator-10 is an orally active, potent positive allosteric modulator (PAM) of the α1β2γ2 GABAA receptor with favorable blood-brain barrier (BBB) penetration. GABAA receptor modulator-10 enhances α1β2γ2 GABAA receptor function and potentiates GABA-evoked currents. GABAA receptor modulator-10 demonstrates potent antiepileptic efficacy in both the Pentetrazol (PTZ) - and Kainic Acid (KA) -induced mice epilepsy models. GABAA receptor modulator-10 can be used for the study of epilepsy[1].
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Molecular Formula
C20H15ClFN5O
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Molecular Weight
395.82
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Smiles
O=C(NC1=CC=C(Cl)C=C1)C2=CC(C3=C4N=CN(CC)C4=NC=N3)=CC=C2F
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Target
GABA Receptor
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Shipping Conditions
Room temperature
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GABAA receptor modulator-10
GABAA receptor modulator-10 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.