GABAA receptor modulator-5 [CAS 3021554-08-2]
GABAA receptor modulator-5 [CAS 3021554-08-2]
SKU:QM-0119598
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Product Details
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Description
GABAA receptor modulator-5 (Compound S28) is a modulator for (γ-aminobutyric acid) A receptor (GABAA receptor), with EC50 of 56 nM and 10 nM, for α1β2γ2 and α4β3δ subtype. GABAA receptor modulator-5 exhibits good pharmacokinetic characteristics in rats. GABAA receptor modulator-5 is slightly toxic toxicity in rats with a loss of rollover reflex (LORR) threshold dose of 23.3 μmol/kg, and exhibits potential ameliorating the postpartum depression[1].
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CAS Number
[3021554-08-2]
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Molecular Formula
C28H36F2N4O3
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Molecular Weight
514.61
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Smiles
C[C@@]12[C@](CC[C@@H]2C(CN3C=NN(C4=CC(F)=NC(F)=C4)C3=O)=O)([H])[C@]5([H])CC[C@]6([H])C[C@@](O)(C)CC[C@]6([H])[C@@]5([H])CC1
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Target
GABA Receptor
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Shipping Conditions
Room temperature
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GABAA receptor modulator-5 [CAS 3021554-08-2]
GABAA receptor modulator-5 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.