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GAK inhibitor 49 [CAS 319492-82-5]
GAK inhibitor 49 [CAS 319492-82-5]
SKU:QM-0077298-01
£363.47 GBP
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Product Details
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Description
GAK inhibitor 49 is a potent, ATP-competitive and highly selective cyclin G associated kinase (GAK) inhibitor with a Ki of 0.54 nM and a cell IC50 of 56 nM. GAK inhibitor 49 also shows binding to RIPK2[1].
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CAS Number
[319492-82-5]
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Molecular Formula
C20H22N2O5
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Molecular Weight
370.4
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Smiles
COC1=C(OC)C(OC)=CC(NC2=CC=NC3=CC(OC)=C(OC)C=C23)=C1
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Target
Cyclin G-associated Kinase (GAK)
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Concentration
10mM
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Purity
98.79
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Solubility
DMSO : 62.5 mg/mL (ultrasonic)
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Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
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Shipping Conditions
Room Temperature
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Hazard Statement
H302, H315, H319, H335
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Precautions
H302, H315, H319, H335
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GAK inhibitor 49 [CAS 319492-82-5]
GAK inhibitor 49 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.