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GCGR antagonist 2 [CAS 280134-25-0]

GCGR antagonist 2 [CAS 280134-25-0]

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QM-0149900-01

£501.98 GBP
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Product Details

  • Description

    GCGR antagonist 2, a Furan-2-carbohydrazide, is an orally active glucagon receptor antagonist. GCGR antagonist 2 binds to hGluR with an Kd value of 2.3 nM, and inhibits rat receptor with an IC50 value of 0.43 nM. GCGR antagonist 2 inhibits glucagon-stimulated glycogenolysis[1][2].

  • CAS Number

    [280134-25-0]

  • Molecular Formula

    C28H26N4O2

  • Molecular Weight

    450.53

  • Smiles

    N#CC1=CC(C(N/N=C/C2=CC=CC3=C2C=CN3CC4=C(C)C(C)=CC(C)=C4C)=O)=CC=C1O

  • Target

    GCGR

  • Purity

    99.76

  • Solubility

    DMSO : 100 mg/mL (ultrasonic)

  • Storage Conditions

    -20°C, 3 years; 4°C, 2 years (Powder)

  • Shipping Conditions

    Room Temperature
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Variant Variant total Quantity Price Variant total
5 mgQM-0149900-01
5 mgQM-0149900-01
£501.98/ea		 £0.00
£501.98/ea £0.00
10 mgQM-0149900-02
10 mgQM-0149900-02
£791.15/ea		 £0.00
£791.15/ea £0.00
25 mgQM-0149900-03
25 mgQM-0149900-03
£1,531.09/ea		 £0.00
£1,531.09/ea £0.00
50 mgQM-0149900-04
50 mgQM-0149900-04
£2,422.89/ea		 £0.00
£2,422.89/ea £0.00
100 mgQM-0149900-05
100 mgQM-0149900-05
£3,840.80/ea		 £0.00
£3,840.80/ea £0.00
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GCGR antagonist 2 [CAS 280134-25-0]

GCGR antagonist 2 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.