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Glucocorticoid receptor modulator 1 [CAS 2868357-11-1]

Glucocorticoid receptor modulator 1 [CAS 2868357-11-1]

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QM-0150685-01

£263.84 GBP
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Product Details

  • Description

    Glucocorticoid receptor modulator 1 is a highly potent and orally active non-steroidal selective glucocorticoid receptor modulator with an IC50 value of 9 nM and 130 nM for NF-κB and AP-1, respectively. Glucocorticoid receptor modulator 1 can effectively reduce the expression of inflammatory factors IL-6, IL-1β, TNF-α, also can relieve dermatitis in mice[1].

  • CAS Number

    [2868357-11-1]

  • Molecular Formula

    C24H23ClN2O4S

  • Molecular Weight

    470.97

  • Smiles

    COC1=C(C=C(C(C)=C1)Cl)S(=O)(NC2=CC=C3C(CCCN3C(C4=CC=CC=C4)=O)=C2)=O

  • Target

    AP-1; Glucocorticoid Receptor; NF-κB

  • Concentration

    10mM

  • Purity

    99.79

  • Solubility

    DMSO : 100 mg/mL (ultrasonic)

  • Storage Conditions

    4°C (Powder, sealed storage, away from moisture and light)

  • Shipping Conditions

    Room Temperature
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Variant Variant total Quantity Price Variant total
5 mgQM-0150685-01
5 mgQM-0150685-01
£263.84/ea		 £0.00
£263.84/ea £0.00
10 mM - 1 mLQM-0150685-02
10 mM - 1 mLQM-0150685-02
£271.13/ea		 £0.00
£271.13/ea £0.00
10 mgQM-0150685-03
10 mgQM-0150685-03
£388.99/ea		 £0.00
£388.99/ea £0.00
25 mgQM-0150685-04
25 mgQM-0150685-04
£727.97/ea		 £0.00
£727.97/ea £0.00
50 mgQM-0150685-05
50 mgQM-0150685-05
£1,035.37/ea		 £0.00
£1,035.37/ea £0.00
100 mgQM-0150685-06
100 mgQM-0150685-06
£1,430.24/ea		 £0.00
£1,430.24/ea £0.00
200 mgQM-0150685-07
200 mgQM-0150685-07
£1,918.67/ea		 £0.00
£1,918.67/ea £0.00
500 mgQM-0150685-08
500 mgQM-0150685-08
£3,564.99/ea		 £0.00
£3,564.99/ea £0.00
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Glucocorticoid receptor modulator 1 [CAS 2868357-11-1]

Glucocorticoid receptor modulator 1 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.