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GnRH-R antagonist 1 [CAS 2826273-90-7]
GnRH-R antagonist 1 [CAS 2826273-90-7]
SKU:QM-0069257
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Product Details
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Description
GnRH-R antagonist 1 (compound 21a) is an orally safe and membrane-permeable GnRH-R antagonist with high binding affinity (IC50=0.57 nM) and potent in vitro antagonistic activity (IC50=2.18 nM) . GnRH-R antagonist 1 can be used in studies of advanced prostate cancer and premature LH peaks preventing[1].
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CAS Number
[2826273-90-7]
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Molecular Formula
C31H28F5N7O6S
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Molecular Weight
721.65
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Smiles
O=C(NOC)NC1=CC=C(C(S2)=C(CN(C)CCOC(F)(F)F)C(C(N3C4=NN=C(OC)C=C4)=O)=C2N(CC5=C(F)C=CC=C5F)C3=O)C=C1
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Target
GnRH Receptor
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Solubility
10 mM in DMSO
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Shipping Conditions
Room temperature
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GnRH-R antagonist 1 [CAS 2826273-90-7]
GnRH-R antagonist 1 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.