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GPR183 antagonist-3
GPR183 antagonist-3
SKU:QM-0135628-01
£269.91 GBP
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Product Details
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Description
GPR183 antagonist-3 (compound 33) is an oral active GPR183 antagonist with the IC50 of 8.7 μM. GPR183 antagonist-3 displays strong in vitro antimigration and anti-inflammatory activity in monocytes, and improves the pathological symptoms of DSS-induced experimental colitis[1].
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Molecular Formula
C21H19BrN4O2S
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Molecular Weight
471.37
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Smiles
BrC1=CC=C(C=C1)/C=C/C(N2CCN(CC2)C(C3=CC=C4N=C(SC4=C3)N)=O)=O
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Target
EBI2/GPR183
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Purity
98.79
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Solubility
DMSO : 100 mg/mL (ultrasonic)
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Storage Conditions
4°C (Powder, protect from light)
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Shipping Conditions
Room Temperature
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GPR183 antagonist-3
GPR183 antagonist-3 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.