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GPR81 agonist 1 [CAS 1620992-67-7]

GPR81 agonist 1 [CAS 1620992-67-7]

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QM-0145315-01

£551.80 GBP
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Product Details

  • Description

    GPR81 agonist 1 is a potent and highly selective GPR81 agonist, with EC50s of 58 nM and 50 nM for human and mouse GPR81, respectively. GPR81 agonist 1 inhibits lipolysis in differentiated 3T3-L1 adipocytes. GPR81 agonist 1 suppresses lipolysis in mice without cutaneous flushing. GPR81 agonist 1 displays remarkable selectivity for GPR81 over GPR109a[1].

  • CAS Number

    [1620992-67-7]

  • Molecular Formula

    C22H30N4O2S2

  • Molecular Weight

    446.63

  • Smiles

    O=C([C@H]1CC[C@H](C)CC1)NC2=NC(C3=CC=CS3)=C(CC(N4CCN(C)CC4)=O)S2

  • Target

    Hydroxycarboxylic Acid Receptor (HCAR)

  • Isoform

    HCAR1

  • Purity

    99.73

  • Solubility

    DMSO : 50 mg/mL (ultrasonic)

  • Storage Conditions

    -20°C, 3 years; 4°C, 2 years (Powder)

  • Shipping Conditions

    Room Temperature
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Variant Variant total Quantity Price Variant total
5 mgQM-0145315-01
5 mgQM-0145315-01
£551.80/ea		 £0.00
£551.80/ea £0.00
10 mM - 1 mLQM-0145315-02
10 mM - 1 mLQM-0145315-02
£602.83/ea		 £0.00
£602.83/ea £0.00
10 mgQM-0145315-03
10 mgQM-0145315-03
£902.93/ea		 £0.00
£902.93/ea £0.00
50 mgQM-0145315-04
50 mgQM-0145315-04
£2,497.01/ea		 £0.00
£2,497.01/ea £0.00
100 mgQM-0145315-05
100 mgQM-0145315-05
£3,690.14/ea		 £0.00
£3,690.14/ea £0.00
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GPR81 agonist 1 [CAS 1620992-67-7]

GPR81 agonist 1 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.