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GRK2 Inhibitor 1 [CAS 24269-96-3]

GRK2 Inhibitor 1 [CAS 24269-96-3]

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QM-0140892-01

£238.32 GBP
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Product Details

  • Description

    GRK2 Inhibitor 1 (methyl 5-[2- (5-nitro-2-furyl) vinyl]-2-furoate) is a dual GRK2/β-ARK1 inhibitor that induces dopamine (DA) inhibition reversal (DIR) . GRK2 Inhibitor 1 can also block serotonin-induced or neurotensin-induced DIR reversal. Note: DIR refers to the phenomenon in which neurons in addiction-related brain pathways become less sensitive to DA inhibition when exposed to moderate concentrations of DA for a long time[1].

  • CAS Number

    [24269-96-3]

  • Molecular Formula

    C12H9NO6

  • Molecular Weight

    263.2

  • Smiles

    O=C(OC)C1=CC=C(O1)/C=C/C2=CC=C(O2)[N+]([O-])=O

  • Target

    Dopamine Receptor; G Protein-coupled Receptor Kinase (GRK)

  • Isoform

    GRK2

  • Purity

    98.06

  • Solubility

    DMSO : 41.67 mg/mL (ultrasonic; warming; heat to 60°C)

  • Storage Conditions

    -20°C, 3 years; 4°C, 2 years (Powder)

  • Shipping Conditions

    Room Temperature

  • Hazard Statement

    H302, H315, H319

  • Precautions

    H302, H315, H319
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Variant Variant total Quantity Price Variant total
5 mgQM-0140892-01
5 mgQM-0140892-01
£238.32/ea		 £0.00
£238.32/ea £0.00
10 mM - 1 mLQM-0140892-02
10 mM - 1 mLQM-0140892-02
£256.55/ea		 £0.00
£256.55/ea £0.00
10 mgQM-0140892-03
10 mgQM-0140892-03
£363.47/ea		 £0.00
£363.47/ea £0.00
25 mgQM-0140892-04
25 mgQM-0140892-04
£740.12/ea		 £0.00
£740.12/ea £0.00
50 mgQM-0140892-05
50 mgQM-0140892-05
£1,116.77/ea		 £0.00
£1,116.77/ea £0.00
100 mgQM-0140892-06
100 mgQM-0140892-06
£1,744.92/ea		 £0.00
£1,744.92/ea £0.00
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GRK2 Inhibitor 1 [CAS 24269-96-3]

GRK2 Inhibitor 1 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.