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GRPR antagonist-1 [CAS 3052544-28-9]
GRPR antagonist-1 [CAS 3052544-28-9]
SKU:QM-0059166
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Product Details
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Description
GRPR antagonist-1 is a potent gastrin releasing peptide receptor (GRPR) antagonist, having the cytotoxicity against certain cancer cells (IC50 of 4.97, 4.36 and 3.40 μM in PC3, Pan02 and HGC-27 cells, respectively) . GRPR antagonist-1 inhibits HGC-27 cell viability by decreasing the Bcl-2 level and increasing the Bax level, causing apoptosis, with anticancer activity[1].
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CAS Number
[3052544-28-9]
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Molecular Formula
C29H33F3N4O4
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Molecular Weight
558.59
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Smiles
CC(C)(OC(N1CCN(CC1)C([C@H](CC2=CNC3=C2C=CC=C3)NC(CC4=CC=C(C=C4)C(F)(F)F)=O)=O)=O)C
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Target
Bombesin Receptor
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Solubility
10 mM in DMSO
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Shipping Conditions
Room temperature
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GRPR antagonist-1 [CAS 3052544-28-9]
GRPR antagonist-1 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.