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GRPR antagonist-3 [CAS 2077238-49-2]
GRPR antagonist-3 [CAS 2077238-49-2]
SKU:QM-0016343
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Product Details
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Description
GRPR antagonist-3 (compound (S) -1m) is a potent GRPR antagonist with an IC50 of 121 nM. GRPR antagonist-3 is stable in rat plasma and towards microsomal oxidative metabolism in vitro. GRPR antagonist-3 can be radiolabeled with fluorine-18 for PET imaging[1].
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CAS Number
[2077238-49-2]
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Molecular Formula
C33H37FN6O5
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Molecular Weight
616.68
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Smiles
O=C(NC1=CC=C(C=C1)[N+]([O-])=O)N[C@](CC2=CNC3=CC=CC=C23)(C)C(NCC4(C5=CC=C(C=N5)OCCF)CCCCC4)=O
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Target
Bombesin Receptor
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Shipping Conditions
Room temperature
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GRPR antagonist-3 [CAS 2077238-49-2]
GRPR antagonist-3 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.