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H3R antagonist 2 [CAS 2970985-05-6]
H3R antagonist 2 [CAS 2970985-05-6]
SKU:QM-0066825
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Product Details
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Description
H3R antagonist 2 (Compound 23) is a multitarget histamine H3 receptor (H3R) antagonist with a Ki of 170 nM for hH3R . H3R antagonist 2 shows inhibitory effects with IC50 values of 180, 880 and 775 nM for acetylcholinesterase, butyrylcholinesterase and human monoamine oxidase B (hMAO B), respectively. H3R antagonist 2 shows favorable anti-neuropathic pain and memory-enhancing effects. H3R can across BBB[1].
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CAS Number
[2970985-05-6]
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Molecular Formula
C24H29NO3
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Molecular Weight
379.49
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Smiles
O=C1C2=CC(OCCCCCN3CCCCCC3)=CC=C2OC4=C1C=CC=C4
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Target
Cholinesterase (ChE) ; Histamine Receptor; Monoamine Oxidase
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Isoform
H3 Receptor; MAO-B
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Solubility
10 mM in DMSO
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Shipping Conditions
Room temperature
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H3R antagonist 2 [CAS 2970985-05-6]
H3R antagonist 2 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.