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H4R antagonist 1 [CAS 1429375-54-1]
H4R antagonist 1 [CAS 1429375-54-1]
SKU:QM-0137101-01
£727.97 GBP
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Product Details
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Description
H4R antagonist 1 is a potent and highly selective histamine H4 receptor (H4R) antagonist with an IC50 of 27 nM. H4R antagonist 1 does not show any noticeable binding affinity to other subtypes of histamine receptors, H1R, H2R, and H3R[1].
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CAS Number
[1429375-54-1]
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Molecular Formula
C11H11BrN8
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Molecular Weight
335.16
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Smiles
CNC(C1)CN1C2=NC3=NC=C(Br)C=C3N4C2=NN=N4
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Target
Histamine Receptor
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Isoform
H4 Receptor
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Concentration
10mM
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Purity
99.82
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Solubility
DMSO : 20 mg/mL (ultrasonic; warming; heat to 60°C)
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Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
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Shipping Conditions
Room Temperature
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H4R antagonist 1 [CAS 1429375-54-1]
H4R antagonist 1 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.