HA2A/hCA XII modulator 1 [CAS 2548963-55-7]
HA2A/hCA XII modulator 1 [CAS 2548963-55-7]
SKU:QM-0067149
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Product Details
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Description
HA2A/hCA XII modulator 1 (compound 14), a triazolopirazine, is a potent hA2A adenosine receptor (hA2AAR) antagonist with Kis of 6.4 nM, 4.819 μM, >30 μM for hA2AAR, hA1AR, hA3AR, respectively. hA2A/hCA XII modulator 1 is a potent human carbonic anhydrase XII (hCA XII) inhibitor with Kis of 6.2 nM, 46 nM, 466 nM, 8.351 μM for hCA XII, hCA II, hCA IX and hCA I, respectively. hA2A/hCA XII modulator 1 has the potential for cancer research[1].
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CAS Number
[2548963-55-7]
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Molecular Formula
C24H19N7O4S
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Molecular Weight
501.52
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Smiles
O=C(NC1=CC=C(C2=CN3C(C(N)=N2)=NN(C4=CC=CC=C4)C3=O)C=C1)C5=CC=C(S(=O)(N)=O)C=C5
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Target
Adenosine Receptor; Carbonic Anhydrase
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Isoform
Adenosine A1 receptor (A1R) ; Adenosine A2A receptor (A2AR) ; Adenosine A3 receptor (A3R) ; CA II; CA XII
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Solubility
10 mM in DMSO
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Shipping Conditions
Room temperature
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HA2A/hCA XII modulator 1 [CAS 2548963-55-7]
HA2A/hCA XII modulator 1 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.