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HIV-1 inhibitor-51 [CAS 2834087-82-8]
HIV-1 inhibitor-51 [CAS 2834087-82-8]
SKU:QM-0069850
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Product Details
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Description
HIV-1 inhibitor-51, a non-nucleoside reverse transcriptase inhibitor (NNRTI), exhibits outstanding antiviral activity against WT HIV-1 (IIIB) and a panel of mutant strains. HIV-1 inhibitor-51 has high binding affinity (KD=2.50 μM) and inhibitory activity (IC50=0.03 μM) to WT HIV-1 RT. HIV-1 inhibitor-51 has EC50s of 2.22-53.3 nM for mutant strains (L100I, K103N, Y181C, Y188L, E138K, F227L + V106A, RES056) [1].
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CAS Number
[2834087-82-8]
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Molecular Formula
C24H19ClFN5O2
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Molecular Weight
463.89
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Smiles
FC(C=C1NC2=NC(OC3=C(C=C(C=C3C)/C=C/C#N)C)=C4C(COC4)=N2)=C(C=C1)C#N.Cl
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Target
HIV; Reverse Transcriptase
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Isoform
HIV-1
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Solubility
10 mM in DMSO
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Shipping Conditions
Room temperature
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HIV-1 inhibitor-51 [CAS 2834087-82-8]
HIV-1 inhibitor-51 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.