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HMCH-1R antagonist 1 [CAS 353487-64-6]
HMCH-1R antagonist 1 [CAS 353487-64-6]
SKU:QM-0097190
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Product Details
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Description
HMCH-1R antagonist 1 (Compound 30) is an effective and selective antagonist of human melanin-concentrating hormone receptor 1 (hMCHR1) with an KB value of 3.6 nM. HMCH-1R antagonist 1 can bind to hMCHR1 and hMCHR2 with IC50 values of 65 nM and 49 nM, respectively. HMCH-1R antagonistist 1 can be used for metabolic research[1].
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CAS Number
[353487-64-6]
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Molecular Formula
C49H82N16O11S3
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Molecular Weight
1167.47
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Smiles
O=C([C@@H](NC([C@@H](NC(CCCCNC([C@@H](NC([C@H](CSSC[C@H](NC(CCCCNC1=O)=O)C(N)=O)NC([C@@H](NC(C)=O)CCCNC(N)=N)=O)=O)CCSC)=O)=O)CCCNC(N)=N)=O)C(C)C)N[C@H]1CC2=CC=C(C=C2)O
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Target
MCHR1 (GPR24)
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Solubility
10 mM in DMSO
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Shipping Conditions
Room temperature
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HMCH-1R antagonist 1 [CAS 353487-64-6]
HMCH-1R antagonist 1 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.