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HTR2A antagonist 1
HTR2A antagonist 1
SKU:QM-0008499
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Product Details
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Description
HTR2A antagonist 1 (Compound 15f) is a HTR2A antagonist, with an IC50 of 42.79 nM. HTR2A antagonist 1 induces sub-G1 cell cycle arrest and apoptosis in colorectal cancer cells via the activation of p53/p21/caspase 3 signaling. HTR2A antagonist 1 has good liver microsomal stability. HTR2A antagonist 1 can be used for the research of colorectal cancer[1].
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Molecular Formula
C35H43Cl2F2N5O4
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Molecular Weight
706.65
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Smiles
O=C(NCC1=CC=C(OCC(O)CN2CCC(C3=NOC4=CC(F)=CC=C34)CC2)C=C1)N(CC5=CC=C(F)C=C5)C6CCNCC6.Cl.Cl
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Target
5-HT Receptor; Apoptosis
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Shipping Conditions
Room temperature
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HTR2A antagonist 1
HTR2A antagonist 1 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.