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I2-IRs ligand-1
I2-IRs ligand-1
SKU:QM-0009773
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Product Details
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Description
I2-IRs ligand-1 (Compound 12d) is an orally active and BBB-penetrable compound. I2-IRs ligand-1 has a high affinity for imidazoline I2 receptors (I2-IRs) (pKi: 9.98) . I2-IRs ligand-1 can improve cognitive impairment in senescent mice and exhibits analgesic, anti-inflammatory, and neuroprotective activities. I2-IRs ligand-1 can be used for the research of Alzheimer's disease and related pain disorders[1].
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Molecular Formula
C21H23ClFN2O4P
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Molecular Weight
452.84
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Smiles
O=C([C@H]1[C@](C2=CC=CC=C2)(P(OCC)(OCC)=O)N=CC1)NC3=CC=C(F)C(Cl)=C3
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Target
Imidazoline Receptor
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Shipping Conditions
Room temperature
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I2-IRs ligand-1
I2-IRs ligand-1 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.