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K-Opioid receptor agonist-1 [CAS 1816990-29-0]
K-Opioid receptor agonist-1 [CAS 1816990-29-0]
SKU:QM-0153024
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Product Details
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Description
K-Opioid receptor agonist-1 (Compound 5a) is an agonist for κ-Opioid receptor with Ki of 0.25 nM and EC50 of 2 nM. K-Opioid receptor agonist-1 is blood brain barrier (BBB) penetrate (brain/plasma ratios of 0.50 to 0.65). K-Opioid receptor agonist-1 exhibits anti-inflammatory activity in dermatitis models induced by Arachidonic acid or oxazolidinone[1].
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CAS Number
[1816990-29-0]
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Molecular Formula
C22H29Cl2N3O3
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Molecular Weight
454.39
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Smiles
ClC(C=C1CC(N2[C@@]3([H])[C@@](CCC[C@@H]3N4CCCC4)([H])N(CC2)C(OC)=O)=O)=C(C=C1)Cl
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Target
Opioid Receptor
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Isoform
δ Opioid Receptor/DOR; κ Opioid Receptor/KOR; μ Opioid Receptor/MOR
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Shipping Conditions
Room temperature
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K-Opioid receptor agonist-1 [CAS 1816990-29-0]
K-Opioid receptor agonist-1 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.