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KOR agonist 2 [CAS 3050912-29-0]

KOR agonist 2 [CAS 3050912-29-0]

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SKU:QM-0080021

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  • Description

    KOR agonist 2 (Compound 23p) is an agonist for κ opioid receptor (KOR) with Ki of 1.9 nM. KOR agonist 2 exhibits analgesic effect in mouse models with ED50 of 1.30 mg/kg. KOR agonist 2 exhibits high clearance rate (2 mg/kg, i.v.) in mice, high metabolism and clearance in liver microsomes[1].

  • CAS Number

    [3050912-29-0]

  • Molecular Formula

    C29H35ClN2O4S

  • Molecular Weight

    543.12

  • Smiles

    O=S(C1=CC=CC(Cl)=C1)(N(CC2=CC=CC=C2)[C@@H]3C[C@H](CN(C)C)[C@](C4=CC=CC(OC)=C4)(O)CC3)=O

  • Target

    Opioid Receptor

  • Isoform

    κ Opioid Receptor/KOR

  • Shipping Conditions

    Room temperature

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KOR agonist 2 [CAS 3050912-29-0]

KOR agonist 2 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.