KOR agonist 4
KOR agonist 4
SKU:QM-0009756
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Product Details
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Description
KOR agonist 4 (compound 39) is an agonist of Kappa Opioid Receptor. KOR agonist 4 is an activator of G-protein signaling. KOR agonist 4 binds with GTPγS with an EC50 of 14 nM and with an Emax of 83 %. KOR agonist 4 demonstrates moderate to high intrinsic clearance in human hepatocytes. KOR agonist 4 exhibits 60- and 810-fold selectivities versus the related mu (MOR) and delta (DOR) opioid receptors. KOR agonist 4 is potential for central nervous system (CNS) disorders research[1].
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Molecular Formula
C21H25N3
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Molecular Weight
319.44
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Smiles
C1(C=C(CCN(CC2CC2)CCC3=CC=CC=C3)C=C4)=C4N=CN1
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Target
Opioid Receptor
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Isoform
δ Opioid Receptor/DOR; κ Opioid Receptor/KOR; μ Opioid Receptor/MOR
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Shipping Conditions
Room temperature
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KOR agonist 4
KOR agonist 4 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.