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M3/PDE4 modulator-1
M3/PDE4 modulator-1
SKU:QM-0072059
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Product Details
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Description
M3/PDE4 modulator-1 (compound 10f) is a bifunctional molecule that is an M3 mAChR antagonist and a PDE4 inhibitor. M3/PDE4 modulator-1 (10-1000 nM/kg; iv) reduces cysteine eosinophil influx in the OVA rat model[1].
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Molecular Formula
C38H41Cl2N3O8S
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Molecular Weight
770.72
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Smiles
COC1=C(OCC)C=C([C@@H](OC(C2=CC=C(CN[C@](C(O[C@H]3CN4CCC3CC4)=O)(CO)C5=CC=CC=C5)S2)=O)CC6=C(Cl)C=[N+]([O-])C=C6Cl)C=C1
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Target
MAChR; Phosphodiesterase (PDE)
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Solubility
10 mM in DMSO
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Shipping Conditions
Room temperature
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M3/PDE4 modulator-1
M3/PDE4 modulator-1 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.