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MOR modulator-1 [CAS 2976336-81-7]

MOR modulator-1 [CAS 2976336-81-7]

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SKU:QM-0009315

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  • Description

    MOR modulator-1 (compound 6) is a potent and selective μ opioid receptor (MOR) modulator. MOR modulator-1 exhibits improved opioid receptor selectivity, enhanced in vivo antagonistic effect, and overall fewer withdrawal symptoms compared to NAT (6α-configuration) . MOR modulator-1 links with carboxamido linker μ, δ, γ with Kis of 0.25, 41.1, 1.30 nM, respectively[1]

  • CAS Number

    [2976336-81-7]

  • Molecular Formula

    C24H27N3O4S

  • Molecular Weight

    453.55

  • Smiles

    O[C@]12[C@@]34C5=C(C[C@@]2([H])N(CC4)CC6CC6)C=CC(O)=C5O[C@@]3([H])[C@H](CC1)NC(C7=NC=CS7)=O

  • Target

    Opioid Receptor

  • Isoform

    δ Opioid Receptor/DOR; κ Opioid Receptor/KOR; μ Opioid Receptor/MOR

  • Shipping Conditions

    Room temperature

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MOR modulator-1 [CAS 2976336-81-7]

MOR modulator-1 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.