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MRGPRX1 agonist 1 [CAS 2377379-39-8]

MRGPRX1 agonist 1 [CAS 2377379-39-8]

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QM-0143061-01

£388.99 GBP
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Product Details

  • Description

    MRGPRX1 agonist 1 is a highly potent MRGPRX1 agonist (EC50=50 nM) with greater than 50-fold selectivity for δ, μ, and κ opioid receptors. MRGPRX1 agonist 1 is inactive against MRGPRC11. MRGPRC11 inhibits high voltage-activated (HVA) Ca2+ currents, reduces neurotransmitter release, and mitigates nociceptive transmission in the spinal cord. MRGPRX1 agonist 1 is useful for the study of chronic pain, especially neuropathic pain[1].

  • CAS Number

    [2377379-39-8]

  • Molecular Formula

    C23H21N3O4S

  • Molecular Weight

    435.5

  • Smiles

    O=S(C1=CC=CC=C1OC)(NC2=CC=C(C)C=C2OC3=CC4=C(C(N)=NC=C4)C=C3)=O

  • Target

    Mas-related G-protein-coupled Receptor (MRGPR)

  • Purity

    99.95

  • Solubility

    DMSO : 125 mg/mL (ultrasonic)

  • Storage Conditions

    -20°C, 3 years; 4°C, 2 years (Powder)

  • Shipping Conditions

    Room Temperature
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Variant Variant total Quantity Price Variant total
5 mgQM-0143061-01
5 mgQM-0143061-01
£388.99/ea		 £0.00
£388.99/ea £0.00
10 mM - 1 mLQM-0143061-02
10 mM - 1 mLQM-0143061-02
£423.00/ea		 £0.00
£423.00/ea £0.00
10 mgQM-0143061-03
10 mgQM-0143061-03
£589.46/ea		 £0.00
£589.46/ea £0.00
25 mgQM-0143061-04
25 mgQM-0143061-04
£1,029.29/ea		 £0.00
£1,029.29/ea £0.00
50 mgQM-0143061-05
50 mgQM-0143061-05
£1,418.09/ea		 £0.00
£1,418.09/ea £0.00
100 mgQM-0143061-06
100 mgQM-0143061-06
£1,970.91/ea		 £0.00
£1,970.91/ea £0.00
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MRGPRX1 agonist 1 [CAS 2377379-39-8]

MRGPRX1 agonist 1 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.