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Mu opioid receptor antagonist 1 [CAS 2767446-03-5]
Mu opioid receptor antagonist 1 [CAS 2767446-03-5]
SKU:QM-0065884
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Product Details
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Description
Mu opioid receptor antagonist 1 (compound 19) is a selective and orally active μ opioid receptor (MOR) ligand with an Ki value of 0.58 nM and an EC50 of 1.15 nM. Orally administrating with Mu opioid receptor antagonist 1 increases intestinal motility during morphine-induced constipation. Mu opioid receptor antagonist 1 can be used for researching opioid-induced constipation (OIC) [1].
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CAS Number
[2767446-03-5]
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Molecular Formula
C24H28N4O4
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Molecular Weight
436.5
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Smiles
O[C@]12[C@H]3CC4=C5[C@@]1(CCN3CC6CC6)[C@H]([C@@H](CC2)NC(C7=CN=CN7)=O)OC5=C(O)C=C4
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Target
Opioid Receptor
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Isoform
μ Opioid Receptor/MOR
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Solubility
10 mM in DMSO
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Shipping Conditions
Room temperature
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Mu opioid receptor antagonist 1 [CAS 2767446-03-5]
Mu opioid receptor antagonist 1 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.